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5. Direct Synthesis of 2,3-Diaroyl Quinolines and Pyridazino[4,5-b]quinolines via an I2-Promoted One-Po

Direct Synthesis of 2,3-Diaroyl Quinolines and Pyridazino[4,5-b]quinolines via an I2-Promoted One-Po

来源 :中国化学会第十六届全国有机合成化学学术研讨会 | 被引量 : 0次 | 上传用户：ankang1989

【摘 要】

：

Quinolines are privileged aromatic aza-heterocycles found in wide range of natural product.1 Povarov reaction is the most effective,enabling the rapid assembly of quinolones.However,recent progress in

【作 者】

：

Peng Zhao An-Xin Wu 

【机 构】

：

Key Laboratory of Pesticide & Chemical Biology,Ministry of Education,College of Chemistry,Central Ch

【出 处】

：

中国化学会第十六届全国有机合成化学学术研讨会

【发表日期】

：

2019年3期

【关键词】

：

2 3-Diaroyl Quinolines Pyridazino[4 5-b]quinolines One-Pot synthesis 1 4-dicarbo 

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　　Quinolines are privileged aromatic aza-heterocycles found in wide range of natural product.1 Povarov reaction is the most effective,enabling the rapid assembly of quinolones.However,recent progress in the Povarov reaction has mainly focused on the synthesis of quinolines containing only one carbonyl group.

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