降压宝蓝片含药血清对过氧化氢损伤的人脐静脉内皮细胞的保护作用

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目的:探讨降压宝蓝片含药血清对过氧化氢(H2O2)诱导人脐静脉血管内皮细胞(HUVECs)损伤的保护作用。方法:体外培养HUVECs,分为空白组、模型组、降压宝蓝片含药血清低、中、高浓度组(含量血清体积分数为5%,10%,15%),显微镜下观察细胞形态,用噻唑蓝(MTT)法检测HUVECs活力,微板法检测上清液中乳酸脱氢酶(LDH)的活性及一氧化氮(NO)的含量,ELISA法检测内皮素-1(ET-1),组织型纤溶酶原激活物(t PA),组织型纤溶酶原激活物抑制剂(PAI-1)的含量。结果:与空白组比较,模型组细胞活力显著降低,上清液中LDH活性明显增高,ET-1和PAI-1含量显著增加,NO和t PA含量显著下降(P<0.01);与模型组比较,降压宝蓝片中、高浓度组细胞活力显著升高,LDH活性显著减低,ET-1和PAI-1含量显著减少,NO和t PA显著升高(P<0.05,P<0.01)。结论:降压宝蓝片含药血清对H2O2诱导的HUVECs损伤具有显著地保护作用。 Objective: To investigate the protective effect of Jianbo Bao Lan Tablet containing serum on the injury of human umbilical vein endothelial cells (HUVECs) induced by hydrogen peroxide (H2O2). Methods: HUVECs were cultured in vitro and divided into blank group, model group, Jianbo Bao Lan Tablet containing low, medium and high serum concentration (content of serum volume fraction of 5%, 10%, 15%) under a microscope to observe the cell morphology, The activity of lactate dehydrogenase (LDH) and nitric oxide (NO) in supernatant were detected by MTT assay and the activity of endothelin-1 (ET-1) , Tissue-type plasminogen activator (t PA), tissue-type plasminogen activator inhibitor (PAI-1) content. Results: Compared with the blank group, the viability of model group decreased significantly, the activity of LDH in the supernatant increased significantly, the contents of ET-1 and PAI-1 increased significantly and the content of NO and t PA decreased (P <0.01) Compared with the control group, the cell viability in high concentration group was significantly increased, the LDH activity was significantly decreased, the content of ET-1 and PAI-1 was significantly decreased, NO and t PA were significantly increased (P <0.05, P <0.01). Conclusion: The antihypertensive Baolan tablets containing serum have a significant protective effect on H2O2-induced HUVECs injury.
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